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Eugene C. Chen

Medical College of Wisconsin · US
Area of research
Oncology · Rheumatology
Research interest
Research interests include Drug Transport and Resistance Mechanisms, Folate and B Vitamins Research, Metabolism and Genetic Disorders, and Pharmacological Effects and Toxicity Studies.
h-index
13
citations
841
works
17
NIH funding
primary concept
email

Recent publications

Tissue distribution and retention drives efficacy of rapidly clearing VHL-based PROTACs
Communications Medicine 2024cited by 18position: middledoi
New and Emerging Research on Solute Carrier and ATP Binding Cassette Transporters in Drug Discovery and Development: Outlook From the International Transporter Consortium
Clinical Pharmacology & Therapeutics 2022cited by 47position: middledoi
Organic cation transporter 1 (OCT1) modulates multiple cardiometabolic traits through effects on hepatic thiamine content
PLoS Biology 2018cited by 63position: middledoi
Discovery of Competitive and Noncompetitive Ligands of the Organic Cation Transporter 1 (OCT1; SLC22A1)
Journal of Medicinal Chemistry 2017cited by 64position: firstdoi
Metformin Is a Substrate and Inhibitor of the Human Thiamine Transporter, THTR-2 (SLC19A3)
Molecular Pharmaceutics 2015cited by 108position: middledoi
Targeted Disruption of Organic Cation Transporter 3 Attenuates the Pharmacologic Response to Metformin
Molecular Pharmacology 2015cited by 101position: firstdoi
OCT1 is a high-capacity thiamine transporter that regulates hepatic steatosis and is a target of metformin
Proceedings of the National Academy of Sciences 2014cited by 236position: middledoi

Grants

Collaborative Research: MFS-SPEED: D-Diameter - Data-Driven Innovation Advancing Macromolecular Engineering Towards Efficient Recycling
NSF2517827$1,250,0002025–2028PIRePORTER
CAS: Lewis Pair Polymerization: Compounded Sequence and Spatiotemporal Controls for Precision Synthesis of Sustainable Linear and Cyclic Block Copolymers
NSF2305058$699,2542023–2027PIRePORTER
CAS: Diastereoselective Polymerization Catalysis for Stereo-Sequenced Polymers with Biodegradability and Chemical Circularity
NSF1955482$490,0002020–2024PIRePORTER
Lewis Pair Polymerization: Controlling Polymer Tacticity and Topology
NSF1904962$664,2502019–2023PIRePORTER
SusChEM: Stereoselective Polymerization Catalysis of Biomass Monomers by Chiral Transition-Metal and Organic Catalysts
NSF1664915$450,0002017–2020PIRePORTER
SusChEM: Lewis Pair Polymerization: A Powerful Synthetic Strategy for Sustainable and Functional Polymers
NSF1507702$540,0002015–2019PIRePORTER
SusChEM: Stereoselective Polymerization of Biomass Monomers by Transition-Metal and Organic Catalysts
NSF1300267$447,0002013–2016PIRePORTER
Synthesis of Sustainable Polymers by Silylium-Catalyzed Polymerization of Renewable Feedstocks
NSF1150792$386,1272012–2015PIRePORTER
Asymmetric Coordination Polymerization Catalysis of Polar Vinyl Monomers
NSF1012326$420,0002010–2013PIRePORTER
Asymmetric Catalysis by Chiral-Polymer-Induced and Stabilized, Chiral-Surface Nanoclusters
NSF0756633$400,0002009–2012PIRePORTER
Living and Stereoselective Anionic Polymerization by Dinuclear Ambiphilic Silicon Propagators
NSF0848845$260,0002009–2012PIRePORTER
Diastereospecific Ion-Pairing Polymerization of Functionalized Vinyl Monomers
NSF0718061$448,0002007–2010PIRePORTER
SBIR Phase I: Exchange Coupling Enabled Scalable High Density Nonvolatile STT-RAM at Fast Speed and Low Power
NSF0711564$99,9932007–2007PIRePORTER
Diastereospecific Ion-Pairing, "Amphicatalytic" Polymerization of Functionalized Vinyl Monomers
NSF0415270$384,0002004–2007PIRePORTER

Frequent collaborators

Kathleen M. Giacomini · University of California, San Francisco6 papers (2014–2022)Sook Wah Yee · Pfizer (United States)6 papers (2014–2022)Huan‐Chieh Chien · Amgen (United States)4 papers (2014–2018)Xiaomin Liang · Southwest University4 papers (2014–2017)Ligong Chen · Hebei Agricultural University3 papers (2014–2018)Meiling Piao · Chinese Academy of Sciences2 papers (2015–2018)Ling Zou · Bioanalytica (Switzerland)2 papers (2018–2022)Kari M. Morrissey · Sanofi (United States)1 papers (2014–2014)Xiaomin Liang · Gilead Sciences (United States)1 papers (2018–2018)John Kurhanewicz · University of California, San Francisco1 papers (2014–2014)Andrej Săli · QB31 papers (2017–2017)Frode Norheim · University of Oslo1 papers (2018–2018)Bin Ma · Shandong University1 papers (2024–2024) · 1 papers (2024–2024)S. Cyrus Khojasteh · China Pharmaceutical University1 papers (2024–2024)Adrian S. Ray · Gilead Sciences (United States)1 papers (2015–2015)Sarah King · University of Queensland1 papers (2018–2018)Jolyn Twelves · Gilead Sciences (United States)1 papers (2015–2015)Shuanglian Li · Children's Hospital of Chongqing Medical University1 papers (2014–2014)Michael J. Lin · University of California, San Francisco1 papers (2014–2014)