Area of research
Infectious Diseases · Molecular Biology
Research interest
Research interests include Chemistry, Mycobacterium tuberculosis, Moiety, In vivo, Antimycobacterial, and Tuberculosis.
Design, synthesis and antimycobacterial activity of novel benzothiazinones with improved water solubility
Design, synthesis and antitubercular activity of novel N-(amino)piperazinyl benzothiazinones with improved safety
Human antibodies targeting a Mycobacterium transporter protein mediate protection against tuberculosis
Design, synthesis and biological activity of N-(amino)piperazine-containing benzothiazinones against Mycobacterium tuberculosis
Design, synthesis and biological evaluation of nitrofuran-1,3,4-oxadiazole hybrids as new antitubercular agents
Design, synthesis and antimycobacterial activity of new benzothiazinones inspired by rifampicin/rifapentine
Identification of benzothiazinones containing an oxime functional moiety as new anti-tuberculosis agents
hERG optimizations of IMB1603, discovery of alternative benzothiazinones as new antitubercular agents
Primary Clofazimine and Bedaquiline Resistance among Isolates from Patients with Multidrug-Resistant Tuberculosis
<i>In Vitro</i> and <i>In Vivo</i> Activities of the Nitroimidazole TBA-354 against Mycobacterium tuberculosis