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Leslie Z. Benet

City College of San Francisco · US
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Area of research
Oncology · Pharmacology
Research interest
Research interests include Drug Transport and Resistance Mechanisms, Pharmacogenetics and Drug Metabolism, Pharmacological Effects and Toxicity Studies, and Analytical Methods in Pharmaceuticals.
h-index
89
citations
37,766
works
636
NIH funding
primary concept
email

Recent publications

Mathematical Modeling in Drug Metabolism and Pharmacokinetics: Correct In Vitro, Not Always Valid In Vivo
Pharmaceuticals 2026cited by 0position: contributordoi
Application of Kirchhoff’s Laws to pharmacologic and pharmacokinetic analyses
Pharmacological Reviews 2025cited by 5position: contributordoi
Response to the commentary on “are all measures of liver Kpuu a function of FH, as determined following oral dosing, or have we made a critical error in defining hepatic drug clearance?”
European Journal of Pharmaceutical Sciences 2025cited by 3position: contributordoi
Net Influx Rather Than Directional Rates: Re-evaluating Transporter Characterization In Vivo and In Vitro for Renal and Hepatic Clearance
The AAPS Journal 2025cited by 2position: contributordoi
An Explanation of Why Dose-Corrected Area Under the Curve for Alternate Administration Routes Can Be Greater than for Intravenous Dosing
The AAPS Journal 2024cited by 13position: contributordoi
Commentary: Pharmacokinetic Theory Must Consider Published Experimental Data
Drug Metabolism and Disposition 2024cited by 10position: contributordoi
Is there a possibility that P‐glycoprotein reduces reproductive toxicity in males but breast cancer resistance protein does not?
Clinical and Translational Science 2024cited by 0position: contributordoi
The Uses and Advantages of Kirchhoff’s Laws vs. Differential Equations in Pharmacology, Pharmacokinetics, and (Even) Chemistry
The AAPS Journal 2023cited by 17position: contributordoi
Solubility-Permeability Interplay in Facilitating the Prediction of Drug Disposition Routes, Extent of Absorption, Food Effects, Brain Penetration and Drug Induced Liver Injury Potential
Journal of Pharmaceutical Sciences 2023cited by 11position: contributordoi
State of the Art and Uses for the Biopharmaceutics Drug Disposition Classification System (BDDCS): New Additions, Revisions, and Citation References
The AAPS Journal 2022cited by 56position: lastdoi
State of the Art and Uses for the Biopharmaceutics Drug Disposition Classification System (BDDCS): New Additions, Revisions, and Citation References
The AAPS Journal 2022cited by 52position: contributordoi
Using an animal model to predict the effective human dose for oral multiple sclerosis drugs
Clinical and Translational Science 2022cited by 10position: contributordoi
Successful and Unsuccessful Prediction of Human Hepatic Clearance for Lead Optimization
Journal of Medicinal Chemistry 2021cited by 60position: contributordoi
Successful and Unsuccessful Prediction of Human Hepatic Clearance for Lead Optimization
Journal of Medicinal Chemistry 2021cited by 59position: lastdoi
There is Only One Valid Definition of Clearance: Critical Examination of Clearance Concepts Reveals the Potential for Errors in Clinical Drug Dosing Decisions
The AAPS Journal 2021cited by 30position: contributordoi
Investigating Intestinal Transporter Involvement in Rivaroxaban Disposition through Examination of Changes in Absorption
Pharmaceutical Research 2021cited by 12position: contributordoi
Examination of Urinary Excretion of Unchanged Drug in Humans and Preclinical Animal Models: Increasing the Predictability of Poor Metabolism in Humans
Pharmaceutical Research 2021cited by 10position: contributordoi
Analyzing Potential Intestinal Transporter Drug-Drug Interactions: Reevaluating Ticagrelor Interaction Studies
Pharmaceutical Research 2021cited by 10position: contributordoi
Using Individualized Patient Data for Prediction of Population Dosing Recommendations Versus Predictions of Individualized Patient Dosing
The Journal of Clinical Pharmacology 2021cited by 0position: contributordoi
The Critical Role of Passive Permeability in Designing Successful Drugs
ChemMedChem 2020cited by 108position: middledoi
The Critical Role of Passive Permeability in Designing Successful Drugs.
2020cited by 71position: contributordoi
Late-Stage Failures of Monoclonal Antibody Drugs: A Retrospective Case Study Analysis
Pharmacology 2020cited by 58position: lastdoi
Are There Any Experimental Perfusion Data that Preferentially Support the Dispersion and Parallel-Tube Models over the Well-Stirred Model of Organ Elimination?
Drug Metabolism and Disposition 2020cited by 38position: contributordoi
Investigating the Theoretical Basis for In Vitro–In Vivo Extrapolation (IVIVE) in Predicting Drug Metabolic Clearance and Proposing Future Experimental Pathways
The AAPS Journal 2020cited by 32position: contributordoi
Intestinal Efflux Transporters P-gp and BCRP Are Not Clinically Relevant in Apixaban Disposition
Pharmaceutical Research 2020cited by 21position: contributordoi
Volume of Distribution is Unaffected by Metabolic Drug–Drug Interactions
Clinical Pharmacokinetics 2020cited by 17position: contributordoi
The Necessity of Using Changes in Absorption Time to Implicate Intestinal Transporter Involvement in Oral Drug-Drug Interactions
The AAPS Journal 2020cited by 13position: contributordoi
Predicting Interactions between Rifampin and Antihypertensive Drugs Using the Biopharmaceutics Drug Disposition Classification System
Pharmacotherapy: The Journal of Human Pharmacology and Drug Therapy 2020cited by 10position: contributordoi
In Vitro-In Vivo Extrapolation and Hepatic Clearance-Dependent Underprediction
Journal of Pharmaceutical Sciences 2019cited by 62position: lastdoi
The Presence of a Transporter-Induced Protein Binding Shift: A New Explanation for Protein-Facilitated Uptake and Improvement for In Vitro-In Vivo Extrapolation
Drug Metabolism and Disposition 2019cited by 55position: lastdoi

Grants

Pharmacokinetic Studies on Procainamide and Its Metabolites
NSF7610466$3,6001976–1978PIRePORTER

Frequent collaborators

· 32 papers (2019–2026) · 5 papers (2020–2026)Monica Gandhi · Chan Zuckerberg Initiative (United States)4 papers (2016–2018)Christine M. Bowman · VIR Biotechnology (United States)4 papers (2016–2019)Alexander Louie · University of San Francisco3 papers (2016–2017)Catherine A. Koss · University of California, San Francisco3 papers (2017–2018)Howard Horng · University of California, San Francisco3 papers (2016–2017)Albert Liu · San Francisco Department of Public Health3 papers (2016–2017)Peter Bacchetti · University of California, San Francisco3 papers (2017–2018)Tudor I. Oprea · University of New Mexico3 papers (2012–2022)Adam Frymoyer · Stanford Medicine2 papers (2012–2013)Nageshwar Budha · Amgen (United States)2 papers (2012–2013)Li Di · Air Force Medical University2 papers (2020–2020) · 2 papers (2012–2013)Wei Liu · Elsevier, Inc.2 papers (2020–2024)Suodi Zhai · Peking University2 papers (2020–2024)Mark J. Dresser · Gilead Sciences (United States)2 papers (2012–2013)Rosa H. M. Chan · City University of Hong Kong2 papers (2015–2017)David V. Glidden · San Francisco General Hospital2 papers (2016–2017)Dolly A. Parasrampuria · Astellas Pharma (United States)2 papers (2014–2018)
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