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Zhongxia Zhou

Shandong University · CN
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Area of research
Infectious Diseases · Pulmonary and Respiratory Medicine
Research interest
Research focused on Human immunodeficiency virus (HIV) and Reverse transcriptase, with related work in Mutant, Triazole, Stereochemistry. Notable publications include 'Design, Synthesis, and Evaluation of Thiophene[3,2- d ]pyrimidine Derivatives as HIV-1 Non-nucleoside Reverse Transcriptase Inhibitors with Significantly Improved Drug Resistance...', 'Structure-Based Optimization of Thiophene[3,2- d ]pyrimidine Derivatives as Potent HIV-1 Non-nucleoside Reverse Transcriptase Inhibitors with Improved Potency against...', and 'First discovery of novel 3-hydroxy-quinazoline-2,4(1H,3H)-diones as specific anti-vaccinia and adenovirus agents via ‘privileged scaffold’ refining approach'.
h-index
citations
469
works
9
NIH funding
primary concept
email

Recent publications

Identification of key genes and infiltrating immune cells among acetaminophen-induced acute liver failure and HBV-associated acute liver failure
Annals of Translational Medicine 2022cited by 9position: middledoi
Targeting the hydrophobic channel of NNIBP: discovery of novel 1,2,3-triazole-derived diarylpyrimidines as novel HIV-1 NNRTIs with high potency against wild-type and K103N mutant virus
Organic & Biomolecular Chemistry 2019cited by 48position: firstdoi
Serum heart-type fatty acid-binding protein as a predictor for the development of sepsis-associated acute kidney injury
Expert Review of Molecular Diagnostics 2019cited by 9position: middledoi
Discovery of Novel Diarylpyrimidine Derivatives as Potent HIV-1 NNRTIs Targeting the “NNRTI Adjacent” Binding Site
ACS Medicinal Chemistry Letters 2018cited by 40position: middledoi
Structure-Based Optimization of Thiophene[3,2-<i>d</i>]pyrimidine Derivatives as Potent HIV-1 Non-nucleoside Reverse Transcriptase Inhibitors with Improved Potency against Resistance-Associated Variants
Journal of Medicinal Chemistry 2017cited by 91position: middledoi
Discovery of uracil-bearing DAPYs derivatives as novel HIV-1 NNRTIs via crystallographic overlay-based molecular hybridization
European Journal of Medicinal Chemistry 2017cited by 41position: middledoi
Design, Synthesis, and Evaluation of Thiophene[3,2-<i>d</i>]pyrimidine Derivatives as HIV-1 Non-nucleoside Reverse Transcriptase Inhibitors with Significantly Improved Drug Resistance Profiles
Journal of Medicinal Chemistry 2016cited by 135position: middledoi
First discovery of novel 3-hydroxy-quinazoline-2,4(1H,3H)-diones as specific anti-vaccinia and adenovirus agents via ‘privileged scaffold’ refining approach
Bioorganic & Medicinal Chemistry Letters 2016cited by 50position: middledoi
Discovery of 2-pyridone derivatives as potent HIV-1 NNRTIs using molecular hybridization based on crystallographic overlays
Bioorganic & Medicinal Chemistry 2014cited by 46position: middledoi

Grants

No grants ingested yet.

Frequent collaborators

Peng Zhan · Shandong University7 papers (2014–2019)Xinyong Liu · Shandong University7 papers (2014–2019)Christophe Pannecouque · KU Leuven6 papers (2014–2019)Erik De Clercq · KU Leuven6 papers (2014–2019)Dongwei Kang · Shandong University6 papers (2016–2019)Heng Zhang · National University of Singapore5 papers (2016–2018)Xiao Ding · Shandong University3 papers (2016–2018)Boshi Huang · Shandong University3 papers (2016–2017)Zhipeng Huo · Shandong University3 papers (2017–2018)Gaochan Wu · Shandong University3 papers (2017–2019)Dirk Daelemans · KU Leuven3 papers (2016–2018)Haoran Xu · Shandong University2 papers (2016–2017)Zhao Wang · Shandong University2 papers (2018–2019)Huiqing Liu · Shandong University2 papers (2014–2017)Xueyi Lu · Sun Yat-sen University2 papers (2016–2017)Zengjun Fang · Shandong University2 papers (2016–2017)Lieve Naesens · Rega Institute for Medical Research1 papers (2016–2016)Zhenyu Li · Shandong University1 papers (2016–2016)Meng Wang · Tufts University1 papers (2019–2019)Ting Wang · University of Arizona1 papers (2019–2019)
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