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J. Michael McIntosh

Bank for International Settlements · CH
Area of research
Molecular Biology · Cellular and Molecular Neuroscience
Research interest
Research interests include Nicotinic Acetylcholine Receptors Study, Receptor Mechanisms and Signaling, Neurotransmitter Receptor Influence on Behavior, and Ion channel regulation and function.
h-index
82
citations
22,314
works
350
NIH funding
primary concept
email

Recent publications

Selective Inhibition of Rat α7 Nicotinic Acetylcholine Receptors by LvID, a Newly Characterized α4/7-Conotoxin from <i>Conus lividus</i>
Journal of Medicinal Chemistry 2025cited by 2position: middledoi
An N-Terminally Elongated Peptide From Conus rolani Defines a New Class of Ribbon α-Conotoxins Targeting Muscle nAChRs.
2025cited by 1position: contributordoi
Shape-Shifting Conotoxins Reveal Divergent Pore-Targeting Mechanisms in Nicotinic Receptors
2025cited by 0position: contributordoi
Conotoxins Targeting Voltage-Gated Sodium Ion Channels
Pharmacological Reviews 2024cited by 21position: middledoi
Conotoxins Targeting Voltage-Gated Sodium Ion Channels.
2024cited by 18position: contributordoi
αO-Conotoxin GeXIVA[1,2] Reduced Neuropathic Pain and Changed Gene Expression in Chronic Oxaliplatin-Induced Neuropathy Mice Model
Marine Drugs 2024cited by 8position: middledoi
Computational Design of α-Conotoxins to Target Specific Nicotinic Acetylcholine Receptor Subtypes.
2024cited by 5position: contributordoi
Analogs of α-conotoxin PnIC selectively inhibit α7β2- over α7-only subtype nicotinic acetylcholine receptors via a novel allosteric mechanism.
2024cited by 5position: contributordoi
Using Constellation Pharmacology to Characterize a Novel α-Conotoxin from <i>Conus ateralbus</i>.
2024cited by 4position: contributordoi
Nicotinic acetylcholine receptors: Therapeutic targets for novel ligands to treat pain and inflammation
Pharmacological Research 2023cited by 86position: lastdoi
Role of α6-Nicotinic Receptors in Alcohol-Induced GABAergic Synaptic Transmission and Plasticity to Cholinergic Interneurons in the Nucleus Accumbens
Molecular Neurobiology 2023cited by 19position: middledoi
DM506 (3-Methyl-1,2,3,4,5,6-hexahydroazepino[4,5-<i>b</i>]indole fumarate), a Novel Derivative of Ibogamine, Inhibits α7 and α9α10 Nicotinic Acetylcholine Receptors by Different Allosteric Mechanisms
ACS Chemical Neuroscience 2023cited by 14position: middledoi
Comparison of the Anti-inflammatory Properties of Two Nicotinic Acetylcholine Receptor Ligands, Phosphocholine and pCF3-diEPP
Frontiers in Cellular Neuroscience 2022cited by 22position: middledoi
Alkaloid ligands enable function of homomeric human α10 nicotinic acetylcholine receptors
Frontiers in Pharmacology 2022cited by 19position: lastdoi
RgIA4 Prevention of Acute Oxaliplatin-Induced Cold Allodynia Requires α9-Containing Nicotinic Acetylcholine Receptors and CD3+ T-Cells
Cells 2022cited by 16position: lastdoi
Rapid multi-directed cholinergic transmission in the central nervous system
Nature Communications 2021cited by 41position: middledoi
Selective Penicillamine Substitution Enables Development of a Potent Analgesic Peptide that Acts through a Non-Opioid-Based Mechanism
Journal of Medicinal Chemistry 2021cited by 28position: lastdoi
Discovery of Methylene Thioacetal-Incorporated α-RgIA Analogues as Potent and Stable Antagonists of the Human α9α10 Nicotinic Acetylcholine Receptor for the Treatment of Neuropathic Pain
Journal of Medicinal Chemistry 2021cited by 25position: middledoi
Computational and Functional Mapping of Human and Rat α6β4 Nicotinic Acetylcholine Receptors Reveals Species-Specific Ligand-Binding Motifs
Journal of Medicinal Chemistry 2021cited by 15position: lastdoi
Cy3-RgIA-5727 Labels and Inhibits α9-Containing nAChRs of Cochlear Hair Cells
Frontiers in Cellular Neuroscience 2021cited by 13position: lastdoi
Curses or Cures: A Review of the Numerous Benefits Versus the Biosecurity Concerns of Conotoxin Research
Biomedicines 2020cited by 47position: middledoi
The α9α10 nicotinic acetylcholine receptors antagonist α-conotoxin RgIA reverses colitis signs in murine dextran sodium sulfate model
European Journal of Pharmacology 2020cited by 23position: middledoi
Behavioral and Molecular Basis of Cholinergic Modulation of Pain: Focus on Nicotinic Acetylcholine Receptors
Current topics in behavioral neurosciences 2020cited by 20position: middledoi
Rapid ‘multi-directed’ cholinergic transmission at central synapses
2020cited by 5position: contributordoi
Full activation of an α7-α3β4 nicotinic receptor complex avoids receptor desensitization in human chromaffin cells
2020cited by 0position: contributordoi
Overexpression of P2X3 and P2X7 Receptors and TRPV1 Channels in Adrenomedullary Chromaffin Cells in a Rat Model of Neuropathic Pain
International Journal of Molecular Sciences 2019cited by 43position: middledoi
Conopeptides [V11L;V16D]ArIB and RgIA4: Powerful Tools for the Identification of Novel Nicotinic Acetylcholine Receptors in Monocytes
Frontiers in Pharmacology 2019cited by 40position: lastdoi
RgIA4 Accelerates Recovery from Paclitaxel-Induced Neuropathic Pain in Rats
Marine Drugs 2019cited by 35position: lastdoi
SLPI Inhibits ATP-Mediated Maturation of IL-1β in Human Monocytic Leukocytes: A Novel Function of an Old Player
Frontiers in Immunology 2019cited by 34position: middledoi
Photoactivatable drugs for nicotinic optopharmacology
Nature Methods 2018cited by 56position: middledoi

Grants

Improvements In Radiocarbon And Archaeomagnetism Dating Techniques
NSF1534094$86,4192015–2018PIRePORTER
Doctoral Dissertation Improvement Grant: Social and Political Interaction in South Africa
NSF1058306$20,0002010–2012PIRePORTER
Archaeological Investigations in the Inland Niger Delta, Mali (West Africa)
NSF8004868$78,6011980–1983PIRePORTER

Frequent collaborators

Sean Christensen · University of Utah13 papers (2012–2022)Arik J. Hone · University of Utah12 papers (2013–2023) · 11 papers (2016–2022)Winfried Padberg · Johannes Gutenberg University Mainz10 papers (2016–2022) · 10 papers (2016–2022)Dongting Zhangsun · Ministry of Education of the People's Republic of China9 papers (2012–2025)Maryka Quik · AbbVie (United States)9 papers (2012–2015)David J. Craik · Australian Research Council9 papers (2012–2025) · 8 papers (2020–2025) · 8 papers (2016–2019)Sulan Luo · Ministry of Education of the People's Republic of China8 papers (2012–2025)Xiaopeng Zhu · Guangxi University8 papers (2012–2025) · 7 papers (2016–2019)M. Imad Damaj · Virginia Commonwealth University6 papers (2012–2020) · 6 papers (2017–2018) · 6 papers (2012–2015)Ryan M. Drenan · Wake Forest University6 papers (2013–2018)Joanna Gajewiak · University of Utah6 papers (2013–2021)Yuanyan Hu · Southwest University5 papers (2012–2015)Baldomero M. Olivera · University of Copenhagen5 papers (2013–2021)