Area of research
Molecular Biology · Hematology
Research interest
Research focused on Bromodomain and Combretastatin, with related work in Stereochemistry, CREB-binding protein, Tubulin. Notable publications include 'Design, synthesis, biological evaluation and cocrystal structures with tubulin of chiral β -lactam bridged combretastatin A-4 analogues as potent antitumor agents', 'Discovery of High-Affinity Inhibitors of the BPTF Bromodomain', and 'Discovery of novel CBP bromodomain inhibitors through TR-FRET-based high-throughput screening'.
Discovery of High-Affinity Inhibitors of the BPTF Bromodomain
Design, synthesis, and biological evaluation of tetrahydroquinolin derivatives as potent inhibitors of CBP bromodomain
Discovery of novel CBP bromodomain inhibitors through TR-FRET-based high-throughput screening
Design, synthesis, biological evaluation and cocrystal structures with tubulin of chiral β -lactam bridged combretastatin A-4 analogues as potent antitumor agents